Controlled Dimroth Rearrangement in the Suzuki-Miyaura Cross Coupling of Triazolopyridopyrimidines.
| hal.structure.identifier | Institut de Chimie Organique et Analytique [ICOA] | |
| dc.contributor.author | CHAMPIRÉ, Anthony | |
| hal.structure.identifier | Institut de Chimie Organique et Analytique [ICOA] | |
| dc.contributor.author | VALA, Christine | |
| hal.structure.identifier | Institut de Chimie Organique et Analytique [ICOA] | |
| hal.structure.identifier | Laboratoire de Chimie Biomoléculaires, Substances Naturelles et Réactivité, URAC16 | |
| dc.contributor.author | LAABID, Achraf | |
| hal.structure.identifier | Laboratoire de Chimie Biomoléculaires, Substances Naturelles et Réactivité, URAC16 | |
| dc.contributor.author | BENHARREF, Ahmed | |
| hal.structure.identifier | Institut de Chimie de la Matière Condensée de Bordeaux [ICMCB] | |
| dc.contributor.author | MARCHIVIE, Mathieu | |
| hal.structure.identifier | Institut de Chimie Organique et Analytique [ICOA] | |
| dc.contributor.author | PLÉ, Karen | |
| hal.structure.identifier | Institut de Chimie Organique et Analytique [ICOA] | |
| dc.contributor.author | ROUTIER, Sylvain | |
| dc.date.issued | 2016-12-16 | |
| dc.identifier.issn | 0022-3263 | |
| dc.description.abstractEn | Polynitrogen heterocycles are often subject to Dimroth rearrangement which consists of ring opening, bond rotation, and ring closure. In this note, we report a synthesis of two new families of triazolopyridopyrimidines. Successful functionalization via a Suzuki-Miyaura coupling was performed with total control of triazole (Dimroth) isomerization based on the judicious choice of reaction conditions. | |
| dc.description.sponsorship | Synthèse Organique : des molécules au vivant - ANR-11-LABX-0029 | |
| dc.description.sponsorship | Radiopharmaceutiques Innovants en Oncologie et Neurologie - ANR-11-LABX-0018 | |
| dc.language.iso | en | |
| dc.publisher | American Chemical Society | |
| dc.title.en | Controlled Dimroth Rearrangement in the Suzuki-Miyaura Cross Coupling of Triazolopyridopyrimidines. | |
| dc.type | Article de revue | |
| dc.identifier.doi | 10.1021/acs.joc.6b02357 | |
| dc.subject.hal | Chimie/Matériaux | |
| bordeaux.journal | Journal of Organic Chemistry | |
| bordeaux.page | 12506-12513 | |
| bordeaux.volume | 81 | |
| bordeaux.issue | 24 | |
| bordeaux.peerReviewed | oui | |
| hal.identifier | hal-01432873 | |
| hal.version | 1 | |
| hal.popular | non | |
| hal.audience | Internationale | |
| hal.origin.link | https://hal.archives-ouvertes.fr//hal-01432873v1 | |
| bordeaux.COinS | ctx_ver=Z39.88-2004&rft_val_fmt=info:ofi/fmt:kev:mtx:journal&rft.jtitle=Journal%20of%20Organic%20Chemistry&rft.date=2016-12-16&rft.volume=81&rft.issue=24&rft.spage=12506-12513&rft.epage=12506-12513&rft.eissn=0022-3263&rft.issn=0022-3263&rft.au=CHAMPIR%C3%89,%20Anthony&VALA,%20Christine&LAABID,%20Achraf&BENHARREF,%20Ahmed&MARCHIVIE,%20Mathieu&rft.genre=article |
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