CHAMPIRÉ, Anthony; VALA, Christine; LAABID, Achraf; BENHARREF, Ahmed; MARCHIVIE, Mathieu; PLÉ, Karen; ROUTIER, Sylvain

doi:10.1021/acs.joc.6b02357

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CHAMPIRÉ, Anthony
Institut de Chimie Organique et Analytique [ICOA]

VALA, Christine
Institut de Chimie Organique et Analytique [ICOA]

LAABID, Achraf
Institut de Chimie Organique et Analytique [ICOA]
Laboratoire de Chimie Biomoléculaires, Substances Naturelles et Réactivité, URAC16

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Journal of Organic Chemistry. 2016-12-16, vol. 81, n° 24, p. 12506-12513

American Chemical Society

Resumen en inglés

Polynitrogen heterocycles are often subject to Dimroth rearrangement which consists of ring opening, bond rotation, and ring closure. In this note, we report a synthesis of two new families of triazolopyridopyrimidines. Successful functionalization via a Suzuki-Miyaura coupling was performed with total control of triazole (Dimroth) isomerization based on the judicious choice of reaction conditions.< Leer menos

DOI

http://dx.doi.org/10.1021/acs.joc.6b02357

Proyecto ANR

Synthèse Organique : des molécules au vivant - ANR-11-LABX-0029
Radiopharmaceutiques Innovants en Oncologie et Neurologie - ANR-11-LABX-0018

Orígen

Importado de Hal

Centros de investigación

Institut de Chimie de la Matière Condensée de Bordeaux (ICMCB) - UMR 5026